Release form of the drug Nolvadex on King Pharma – packaging (bank) with 50 tablets each containing 20 mg.
Nolvadex – a brand for products based on the active ingredient tamoxifen citrate. This non-steroidal agent that exhibits antiestrogenic properties. These properties are due to the ability to compete with estrogen substance in different tissues. In medicine, the effect is very useful in the treatment of patients with tumors caused by the action of estrogen. Details.
Bodybuilders, men find Nolvadex very effective in combating the effects of steroids with a strong level of flavoring, resulting in increased levels of estrogen. No compensation or post-cycle therapy (PCT) may develop, such as gynecomastia and the formation of fat deposition, forming a feminine silhouette, and so on. Nolvadex – or rather, Tamoxifen citrate works, occupying estrogen receptors, resulting in the unnecessary use of the drug development of tissues on the chest is significantly reduced and may stop altogether.
The drug is almost non-toxic and has almost no side effects. It fits well with the majority of anabolic cycles, as a counterweight to possible side effects. Note that Nolvadex may slow progress during a steroid cycle. This can be explained by the fact that estrogen plays a role in keeping androgen receptors open. Regardless of this, Nolvadex is the most popular anti-estrogen used male athletes.
Nolvadex working principle
Nolvadex (Tamoxifen Citrate) has no effect on the levels of estrogen in the blood, because its mechanism of action is reduced to blockade the different types of estrogen receptors. Thus, about Tamoxifen citrate can say as not selective (non-selective). Nolvadex binds to estrogen receptors throughout the body. By blocking the receptors throughout the body, it helps to ensure that the body began to rebuild its own testosterone. Importantly, Nolvadex capable of blocking estrogen receptors in the pituitary less than Clomid (Clomid).
Nolvadex reception, assimilation and elimination
If ingestion is rapidly absorbed, and after 5-7 hours in the blood creates a maximum concentration. 99% associated with blood proteins (albumin). Excretion occurs dwuhfazno: Initial T 1/2 from 8 to 14 hours, the final T 1/2 – 7 days.
Start receiving Nolvadex accounts for 2 week steroid cycle, and ends 2-3 weeks after the end of the cycle, the average dose of 10-20 mg per day.
Pay attention to the common misconception that anti-estrogens should be drunk after cycle. This is not true. Estrogen levels rise at the end of the first week of the cycle taking anabolic drugs, so from that moment you need to start taking. If used anabolic drugs that are poorly susceptible aromatization, the need of an aromatase inhibitor during the course eliminated, and tamoxifen citrate Nolvadex activated only at the end of the course. Read more.
This drug is added to the list of banned doping agents. The detection time is 3-6 months depending on the method of detection.